| Name | c Src |
|---|---|
| Synonyms | ASV; SRC1; Avian sarcoma virus protein; Proto oncogene tyrosine protein kinase SRC; SRC; Tyrosine kinase pp60c src; Tyrosine protein kinase SRC 1; c SRC… |
| Name | 4-CPA |
|---|---|
| CAS | 2-(4-chlorophenoxy)acetic acid |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 10819990 | Wang W, Ramdas L, Sun G, Ke S, Obeyesekere NU, Budde RJ, McMurray JS: Cyclic peptides incorporating 4-carboxyphenylalanine and phosphotyrosine are potent inhibitors of pp60 (c-)(src). Biochemistry. 2000 May 2;39(17):5221-8. Of these, 4-carboxyphenylalanine (4-Cpa) and phosphotyrosine resulted in high affinity peptides exhibiting K (i) values of 0.85 and 1.1 microM, respectively, 180- and 130-fold increases in potency over the parent cyclic peptide (K (i) = 150 microM). |
2(0,0,0,2) | Details |