Name | choline esterase |
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Synonyms | Acylcholine acylhydrolase; BCHE; BCHE protein; Butyrylcholine esterase; Butyrylcholinesterase; CHE1; Choline esterase II; Cholinesterase… |
Name | ethephon |
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CAS |
PubMed | Abstract | RScore(About this table) | |
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866390 | Hennighausen G, Tiefenbach B, Lohs Kh: [The effect of 2-chlorethylphosphonic acid (ethephon) on the activity of cholinesterases in vivo and in vitro with reference to its acute toxicity] Pharmazie. 1977 Mar;32(3):181-2. |
6(0,0,1,1) | Details |
9890196 | Sparks SE, Quistad GB, Casida JE: Organophosphorus pesticide-induced butyrylcholinesterase inhibition and potentiation of succinylcholine toxicity in mice. J Biochem Mol Toxicol. 1999;13(2):113-8. The organophosphorus plant defoliant tribufos (4 h pretreatment, 160 mg/kg) and organophosphorus plant growth regulator ethephon (1 h pretreatment, 200 mg/kg) potentiate the toxicity of succinylcholine by seven- and fourfold, respectively. |
5(0,0,0,5) | Details |
727875 | Hennighausen G, Tiefenbach B: [Mechanism of acute toxic effects of chlorocholine and 2-chloroethyl phosphonic acid (Ethephon)]. Arch Exp Veterinarmed. 1978;32(4):609-21. All the cholinesterases studied, including those obtained from plasma, erythrocytes, and brain from rat and mouse, were inhibited in vitro by approximately identical Etephon concentrations. |
1(0,0,0,1) | Details |
18992204 | El-Okazy AM: The Effects of Combination of Ethephon (2-Chloroethyl Phosphonic Acid) (Plant Growth Regulators) on Some Physiological Parameters in Mice. J Egypt Public Health Assoc. 2008;83(1-2):67-86. A highly significant dose dependent variation occurred in acetyl choline esterase (AChE) activity among treated groups. |
- 3 and 1(0,0,0,1) | Details |
10898597 | Haux JE, Quistad GB, Casida JE: Phosphobutyrylcholinesterase: phosphorylation of the esteratic site of butyrylcholinesterase by ethephon [(2-chloroethyl) phosphonic acid] dianion. Chem Res Toxicol. 2000 Jul;13(7):646-51. |
393(4,6,7,8) | Details |
12482234 | Haux JE, Lockridge O, Casida JE: Specificity of ethephon as a butyrylcholinesterase inhibitor and phosphorylating agent. Chem Res Toxicol. 2002 Dec;15(12):1527-33. Butyrylcholinesterase (BChE) is inhibited by the plant growth regulator (2-chloroethyl) phosphonic acid (ethephon) as observed 25 years ago both in vitro and in vivo in rats and mice and more recently in subchronic studies at low doses with human subjects. |
112(1,2,2,2) | Details |
11886791 | Zhang N, Casida JE: Novel irreversible butyrylcholinesterase inhibitors: 2-chloro-1-(substituted-phenyl) ethylphosphonic acids. Bioorg Med Chem. 2002 May;10(5):1281-90. 2-Chloroethylphosphonic acid (ethephon) as the dianion phosphorylates butyrylcholinesterase (BChE) at its active site. |
82(1,1,1,2) | Details |