| Name | alpha adrenoceptors (protein family or complex) |
|---|---|
| Synonyms | Alpha adrenoceptor; Alpha adrenoceptor; Alpha adrenergic receptor; Alpha adrenergic receptors; Alpha adrenoceptors; Alpha adrenoceptors; alpha1 Adrenoceptors; alpha1 Adrenoceptor… |
| Name | tetramine |
|---|---|
| CAS |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 2880286 | Taouis M, Berlan M, Lafontan M: Alpha 2-adrenergic receptor turnover in adipose tissue and kidney: irreversible blockade of alpha 2-adrenergic receptors by benextramine. Mol Pharmacol. 1987 Jan;31(1):89-96. The recovery of post- and extrasynaptic alpha 2-adrenergic receptor-binding sites was studied in vivo in male golden hamsters after treatment with an irreversible alpha-adrenoceptor antagonist benextramine, a tetramine disulfide that possesses a high affinity for alpha 2-binding sites. |
35(0,1,1,5) | Details |
| 6121600 | Belleau B, Benfey BG, Melchiorre C: Presynaptic effect of clonidine antagonized by the tetramine disulphide, benextramine. Br J Pharmacol. 1982 Apr;75(4):617-21. Like phentolamine, benextramine increased the effect of high-voltage stimulation, presumably by blocking presynaptic alpha-adrenoceptors. 3 Clonidine reduced the effect of high-voltage stimulation, presumably by stimulating presynaptic alpha-adrenoceptors. |
2(0,0,0,2) | Details |
| 38001 | Benfey BG, Yong MS, Belleau B, Melchiorre C: Inhibition of the cardiac inotropic effect of by a tetramine disulfide with irreversible alpha-adrenoceptor blocking activity. Can J Physiol Pharmacol. 1979 May;57(5):510-6. BHC was used to test the adrenoceptor interconversion hypothesis which claims that low temperature converts inotropic beta-adrenoceptors in rat atrium and frog ventricle to alpha-adrenoceptors. |
1(0,0,0,1) | Details |
| 6149805 | Vohra MM, Chaudhry A: Antagonism by the tetramine disulfide benextramine of the inhibitory effects mediated by prejunctional alpha 2-adrenoceptors and by postjunctional histamine H2 receptors in the mouse vas deferens. Can J Physiol Pharmacol. 1984 Sep;62(9):1147-51. The actions of benextramine, which blocks postjunctional alpha-adrenoceptors noncompetitively and irreversibly (non-equilibrium type) on prejunctional alpha-adrenoceptors (alpha 2) and postjunctional histamine H2 receptors, were studied in the mouse vas deferens, using clonidine and respectively, as the agonists. |
1(0,0,0,1) | Details |
| 6121599 | Belleau B, Benfey BG, Benfey TJ, Melchiorre C: Inhibition by the tetramine disulphide, benextramine, of cardiac chronotropic histamine H2-receptor-mediated effects. Br J Pharmacol. 1982 Apr;75(4):573-8. |
0(0,0,0,0) | Details |
| 6263429 | Brasili L, Melchiorre C, Belleau B, Benfey BG: Reactivation by of vascular alpha adrenoceptors blocked by the tetramine disulfide benextramine and interaction of benextramine with phenoxybenzamine. Can J Physiol Pharmacol. 1980 Dec;58(12):1490-3. |
82(1,1,1,2) | Details |