| Name | alpha adrenoceptor |
|---|---|
| Synonyms | Alpha 2A Adrenoceptor; ZNF32; ADRA2; ADRA2A; ADRA2R; ADRAR; ALPHA2AAR; Alpha 2A adrenergic receptor… |
| Name | tetramine |
|---|---|
| CAS |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 6113041 | Benfey BG, Belleau B, Brasili L, Giannella M, Melchiorre C: Irreversible alpha adrenoceptor blocking effects and reversible muscarinic blocking and nicotinic blocking effects of tetramine disulfides on the heart. Can J Physiol Pharmacol. 1980 Dec;58(12):1477-83. |
244(3,3,3,4) | Details |
| 34474 | Benfey BG, Yong MS, Belleau B, Melchiorre C: Cardiac muscarinic blocking and atropinic blocking effects of a tetramine disulfide and alpha-adrenoceptor blocking activity. Can J Physiol Pharmacol. 1979 Jan;57(1):41-7. |
162(2,2,2,2) | Details |
| 2871470 | Brasili L, Cassinelli A, Angeli P, Melchiorre C: Thiol group may be involved in the irreversible blockade of presynaptic alpha 2-adrenoreceptors by pyrextramine and benextramine in the isolated guinea pig ileum. Life Sci. 1986 May 5;38(18):1633-40. This study, conducted on isolated guinea pig ileum, was designed to establish the mechanism of presynaptic alpha 2-adrenoreceptor blockade by the tetramine disulfides, benextramine and pyrextramine. |
81(1,1,1,1) | Details |
| 38001 | Benfey BG, Yong MS, Belleau B, Melchiorre C: Inhibition of the cardiac inotropic effect of by a tetramine disulfide with irreversible alpha-adrenoceptor blocking activity. Can J Physiol Pharmacol. 1979 May;57(5):510-6. |
32(0,1,1,2) | Details |
| 2880286 | Taouis M, Berlan M, Lafontan M: Alpha 2-adrenergic receptor turnover in adipose tissue and kidney: irreversible blockade of alpha 2-adrenergic receptors by benextramine. Mol Pharmacol. 1987 Jan;31(1):89-96. The recovery of post- and extrasynaptic alpha 2-adrenergic receptor-binding sites was studied in vivo in male golden hamsters after treatment with an irreversible alpha-adrenoceptor antagonist benextramine, a tetramine disulfide that possesses a high affinity for alpha 2-binding sites. |
31(0,1,1,1) | Details |
| 6121600 | Belleau B, Benfey BG, Melchiorre C: Presynaptic effect of clonidine antagonized by the tetramine disulphide, benextramine. Br J Pharmacol. 1982 Apr;75(4):617-21. 1 The presynaptic alpha-adrenoceptor blocking activity of the newly synthesized alpha-adrenoceptor blocking drug, benextramine, was evaluated in the isolated left atrium of the guinea-pig heart. 2 High-voltage stimulation increased the force of contraction of electrically driven atrial strips, presumably by releasing from sympathetic nerve endings. |
1(0,0,0,1) | Details |