| Name | GRK2 |
|---|---|
| Synonyms | ADRBK 1; ADRBK1; ADRBK1 protein; BARK; BARK 1; BARK1; BETA ARK1; Beta adrenergic receptor kinase 1… |
| Name | chlorpyrifos |
|---|---|
| CAS |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 18800293 | Udarbe Zamora EM, Liu J, Pope CN: Effects of chlorpyrifos oxon on M2 muscarinic receptor internalization in different cell types. J Toxicol Environ Health A. 2008;71(21):1440-7. The active metabolite of the organophosphorus insecticide chlorpyrifos, i.e., chlorpyrifos oxon (CPO), inhibited agonist-induced phosphorylation of human recombinant M2 receptors by GRK2 in vitro in a concentration-dependent manner. |
82(1,1,1,2) | Details |
| 16824341 | Zou LM, Li SY, Zhang J: [Effects of organophosphorus insecticides on G protein-coupled receptor kinase-2 mediated phosphorylation of M2 muscarinic receptors]. Zhonghua Lao Dong Wei Sheng Zhi Ye Bing Za Zhi. 2006 Jun;24(6):352-5. In vitro experiments, the purified mAChR2, G-protein coupled receptor kinase 2 (GRK2) and the (gamma-p32) labeled ATP were incubated with paraoxon (PO), chlorpyrifos oxon (CPO) or chlorpyrifos (CPF) of varying concentrations. |
10(0,0,1,5) | Details |