| Name | Acetylcholinesterases |
|---|---|
| Synonyms | ACHE; ACHE protein; AChE; ARACHE; AcChoEase; Acetylcholine acetylhydrolase; Acetylcholinesterase; Acetylcholinesterase isoform E4 E6 variant… |
| Name | temephos |
|---|---|
| CAS |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 8913110 | Bourguet D, Capela R, Raymond M: An insensitive acetylcholinesterase in Culex pipiens (Diptera:Culicidae) from Portugal. J Econ Entomol. 1996 Oct;89(5):1060-6. Resistance mechanisms of a strain (PRAIAS) of northern house mosquito, Culex pipiens L., collected in Portugal in 1993, and highly resistant to organophosphates and carbamates, were investigated by comparing the resistance characteristics to 3 organophosphorous (temephos, chlorpyrifos, malathion) and 1 (propoxur) insecticides in the presence or absence of synergists; and by determining the possible occurrence of overproduced esterases or insensitive acetylcholinesterase (AChE). |
11(0,0,1,6) | Details |
| 7504077 | Ben Cheikh H, Pasteur N: Resistance to temephos, an organophosphorous insecticide, in Culex pipiens from Tunisia, North Africa. J Am Mosq Control Assoc. 1993 Sep;9(3):335-7. After selecting larvae of one of the samples (ES) with temephos for 6 generations, a 9-fold increase in resistance was observed, and all mosquitoes were found to carry esterases A2-B2 and an insensitive acetylcholinesterase. |
7(0,0,1,2) | Details |
| 10084133 | Wirth MC: Isolation and characterization of two novel organophosphate resistance mechanisms in Culex pipiens from Cyprus. J Am Mosq Control Assoc. 1998 Dec;14(4):397-405. Two strains, one expressing the novel, highly active esterases A5 and B5 (strain A5B5-R), and one expressing insensitive acetylcholinesterase (strain Ace-R), were developed by single pair crosses and selection with temephos and propoxur, respectively. |
7(0,0,1,2) | Details |
| 6193610 | Pellissier C, Leung Tack D, Gras G: [Effect of temephos on acetylcholinesterase activity in the brain of Tilapia guineensis. 3: Comparative effect of temephos and 3 substitute insecticides]. Toxicol Eur Res. 1983 Mar;5(2):63-9. |
7(0,0,1,2) | Details |
| 15115088 | Paeporn P, Komalamisra N, Deesin V, Rongsriyam Y, Eshita Y, Thongrungkiat S: Temephos resistance in two forms of Aedes aegypti and its significance for the resistance mechanism. Southeast Asian J Trop Med Public Health. 2003 Dec;34(4):786-92. The major enzyme-based resistance mechanisms involved in temephos resistance include elevated nonspecific esterase, oxidase and insensitive acetylcholinesterase. |
6(0,0,1,1) | Details |
| 12408646 | Fourcy D, Jumel A, Heydorff M, Lagadic L: Esterases as biomarkers in Nereis (Hediste) diversicolor exposed to temephos and Bacillus thuringiensis var. israelensis used for mosquito control in coastal wetlands of Morbihan (Brittany, France). Mar Environ Res. 2002 Sep-Dec;54(3-5):755-9. Acetylcholinesterase and carboxylesterases were used as biomarkers to assess the effects of Abate 500e (a.i. temephos) and Vectobac 12 AS (a.i. endotoxins of Bacillus thuringiensis var. israelensis, Bti) in Nereis (Hediste) diversicolor. |
6(0,0,1,1) | Details |
| 6189264 | Gras G, Pelissier C, Tack DL: [Effect of temephos on the acetylcholinesterase activity of the brain of Tilapia guineensis. 1: Experimental study at operative doses]. Toxicol Eur Res. 1982 Nov;4(6):301-8. |
6(0,0,1,1) | Details |
| 7514668 | Rivet Y, Raymond M, Rioux JA, Delalbre A, Pasteur N: Resistance monitoring in Culex pipiens (Diptera: Culicidae) from central-eastern France. J Med Entomol. 1994 Mar;31(2):231-9. Insensitive acetylcholinesterase (AceR) and five over-produced esterases (A1, A2 and B2, and A4 and B4) involved in detoxification are responsible for resistance to organophosphorous insecticides (OPs) in Culex pipiens L. from the Rhone-Alpes region, where C. pipiens control is mainly accomplished with the OPs temephos and chlorpyrifos using 0.15 mg/liter doses. |
6(0,0,1,1) | Details |
| 2434168 | Antwi LA: Fish head acetylcholinesterase activity after aerial application of temephos in two rivers in Burkina Faso, West Africa. Bull Environ Contam Toxicol. 1987 Mar;38(3):461-6. |
6(0,0,1,1) | Details |
| 19230585 | Paeporn P, Komalamisra N, Thongrungkiat S, Deesin V, Eshita Y, Rongsriyam Y: Potential development of temephos resistance in Aedes aegypti related to its mechanism and susceptibility to dengue virus. Southeast Asian J Trop Med Public Health. 2003;34 Suppl 2:136-41. The assay for major enzyme-based resistance mechanisms was done in a microtiter plate to detect elevated non-specific esterases, monooxygenase, and insensitive acetylcholinesterase in the temephos-selected and non-selected groups. |
6(0,0,1,1) | Details |
| 6189265 | Pelissier C, Tack DL, Gras G: [Effect of temephos on the acetylcholinesterase activity of the brain of Tilapia guineensis. 2: Experimental study of 24-hour exposure to the toxic compound]. Toxicol Eur Res. 1982 Nov;4(6):309-14. |
6(0,0,1,1) | Details |
| 17915512 | Djogbenou L, Weill M, Hougard JM, Raymond M, Akogbeto M, Chandre F: Characterization of insensitive acetylcholinesterase (ace-1R) in Anopheles gambiae (Diptera: Culicidae): resistance levels and dominance. J Med Entomol. 2007 Sep;44(5):805-10. Furthermore, the dominance status varied between semi-recessivity with fenitrothion and chlorpyrifos methyl insecticides to semidominance with temephos, carbosulfan, and propoxur. |
2(0,0,0,2) | Details |
| 10887565 | Rodriguez MM, Bisset JA, Mila LH, Calvo E, Diaz C, Alain Soca L: [Levels of insecticide resistance and its mechanisms in a strain of Aedes aegypti of Santiago de Cuba]. Rev Cubana Med Trop. 1999 May-Aug;51(2):83-8. The results of bioassays showed low levels of resistance to fention, malathion and deltametrine, moderate levels of resistance to temephos, metyl-pirimifos and cipermetrine and high levels of resistance to chlorpirifios. In accordance with the high frequency values observed in each of the mechanisms, it was proved that esterases and glutathione-S-transferase were involved in the insecticide resistance but acetylcholinesterases were not. |
2(0,0,0,2) | Details |
| 18240518 | Rodriguez MM, Bisset JA, Fernandez D: Levels of insecticide resistance and resistance mechanisms in Aedes aegypti from some Latin American countries. J Am Mosq Control Assoc. 2007 Dec;23(4):420-9. Biochemical tests showed high frequencies of esterase and glutathione-S-transferase activity; however, the frequency of altered acetylcholinesterase mechanism was low. Eight Latin American strains of Aedes aegypti were evaluated for resistance to 6 organophosphates (temephos, malathion, fenthion, pirimiphos-methyl, fenitrothion, and chlorpirifos) and 4 pyrethroids (deltamethrin, lambdacyhalothrin, betacypermethrin, and cyfluthrin) under laboratory conditions. |
1(0,0,0,1) | Details |
| 9439121 | Chandre F, Darriet F, Doannio JM, Riviere F, Pasteur N, Guillet P: Distribution of organophosphate and resistance in Culex pipiens quinquefasciatus (Diptera: Culicidae) in West Africa. J Med Entomol. 1997 Nov;34(6):664-71. For temephos, ratios ranged from 3 to 18 and from 1 to 2, respectively. Cross resistance to organophosphates and carbamates was caused by an insensitive acetylcholinesterase allele (AceR). |
1(0,0,0,1) | Details |
| 9615543 | Ben Cheikh H, Ben Ali-Haouas Z, Marquine M, Pasteur N: Resistance to organophosphorus and pyrethroid insecticides in Culex pipiens (Diptera: Culicidae) from Tunisia. J Med Entomol. 1998 May;35(3):251-60. Resistance to the organophosphates temephos and chlorpyrifos, the propoxur, the pyrethroid permethrin, and the organochloride DDT was investigated in Tunisian populations of Culex pipiens pipiens (L.) collected between 1990 and 1996. To better understand the factors influencing the distribution of resistance in Tunisia, the polymorphism of genes involved in organophosphate resistance (i.e., over-produced esterases and insensitive acetylcholinesterase) was investigated in relation to the genetic structure of populations studied by analyzing the electrophoretic polymorphism of "neutral" genes. |
1(0,0,0,1) | Details |
| 8723267 | Wirth MC, Georghiou GP: Organophosphate resistance in Culex pipiens from Cyprus. J Am Mosq Control Assoc. 1996 Mar;12(1):112-8. All population samples generally revealed organophosphate resistance to malathion, temephos, chlorpyrifos, fenthion, dichlorvos, and pirimiphos methyl, in decreasing order of magnitude. Resistance was associated with the presence of 5 different overproduced esterases (esterases A1, A2, A5, B2, and B5) as well as an insensitive form of acetylcholinesterase. |
1(0,0,0,1) | Details |
| 15311465 | Corbel V, Duchon S, Zaim M, Hougard JM: Dinotefuran: a potential neonicotinoid insecticide against resistant mosquitoes. J Med Entomol. 2004 Jul;41(4):712-7. The results showed that dinotefuran was less toxic than most of the commonly used insecticides (e.g., deltamethrin, carbosulfan, and temephos) against the susceptible mosquitoes tested (between 6- and 100-fold at the LD50 level). More interestingly, the -resistant strain of Cx. quinquefasciatus was significantly more affected by dinotefuran than the susceptible strain (RR = 0.70), probably because the insensitive acetylcholinesterase is less efficient to degrade nicotinic substrates than normal acetylcholinesterase. |
1(0,0,0,1) | Details |
| 17067049 | Zayed AB, Szumlas DE, Hanafi HA, Fryauff DJ, Mostafa AA, Allam KM, Brogdon WG: Use of bioassay and microplate assay to detect and measure insecticide resistance in field populations of Culex pipiens from filariasis endemic areas of Egypt. J Am Mosq Control Assoc. 2006 Sep;22(3):473-82. Microplate assays were performed to measure levels of beta esterase, acetylcholinesterase, insensitive acetylcholinesterase, oxidases, and glutathione-S-transferase enzymes. The Qalubiya larval population was susceptible only to malathion, whereas Sharkiya larvae were susceptible to malathion, temephos, and chlorpyrifos. |
1(0,0,0,1) | Details |
| 10480123 | Pinkney AE, McGowan PC, Murphy DR, Lowe TP, Sparling DW, Meredith WH: Effects of temephos (Abate 4E) on fiddler crabs (Uca pugnax and Uca minax) on a Delaware salt marsh. J Am Mosq Control Assoc. 1999 Sep;15(3):321-9. Median acetylcholinesterase activity in claw muscle of red-jointed fiddler crabs (Uca minax) collected 2 days after an operational spray with Abate 4E was significantly reduced (28% lower) compared to unsprayed crabs. |
1(0,0,0,1) | Details |
| 10480122 | Wirth MC, Georghiou GP: Selection and characterization of temephos resistance in a population of Aedes aegypti from Tortola, British Virgin Islands. J Am Mosq Control Assoc. 1999 Sep;15(3):315-20. |
0(0,0,0,0) | Details |
| 15916049 | Saelim V, Brogdon WG, Rojanapremsuk J, Suvannadabba S, Pandii W, Jones JW, Sithiprasasna R: Bottle and biochemical assays on temephos resistance in Aedes aegypti in Thailand. Southeast Asian J Trop Med Public Health. 2005 Mar;36(2):417-25. |
0(0,0,0,0) | Details |
| 8551300 | Mazzarri MB, Georghiou GP: Characterization of resistance to organophosphate, and pyrethroid insecticides in field populations of Aedes aegypti from Venezuela. J Am Mosq Control Assoc. 1995 Sep;11(3):315-22. Resistance to the organophosphates (OP) temephos, malathion, and pirimiphos methyl, and the propoxur was found to be low (< 5-fold) in 3 Aedes aegypti populations collected from Falcon and Aragua states of Venezuela. |
0(0,0,0,0) | Details |