Name | hormone receptor |
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Synonyms | Early response protein NAK1; GFRP 1; GFRP1; Growth factor inducible nuclear protein N10; Growth factor response protein 1; HMR; Hormone receptor; N10… |
Name | tebufenozide |
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CAS | 3,5-dimethylbenzoic acid 1-(1,1-dimethylethyl)-2-(4-ethylbenzoyl)hydrazide |
PubMed | Abstract | RScore(About this table) | |
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11520684 | Debernard S, Bozzolan F, Duportets L, Porcheron P: Periodic expression of an ecdysteroid-induced nuclear receptor in a lepidopteran cell line (IAL-PID2). Insect Biochem Mol Biol. 2001 Oct;31(11):1057-64. A set of DNA primers was designed within the DNA-binding domain of the Manduca hormone receptor 3 (MHR3) cDNA. |
4(0,0,0,4) | Details |
8763167 | Palli SR, Ladd TR, Sohi SS, Cook BJ, Retnakaran A: Cloning and developmental expression of Choristoneura hormone receptor 3, an ecdysone-inducible gene and a member of the steroid hormone receptor superfamily. Insect Biochem Mol Biol. 1996 May;26(5):485-99. |
3(0,0,0,3) | Details |
9094210 | Palli SR, Ladd TR, Ricci AR, Sohi SS, Retnakaran A: Cloning and development expression of Choristoneura hormone receptor 75: a homologue of the Drosophila E75A gene. Dev Genet. 1997;20(1):36-46. |
2(0,0,0,2) | Details |
12638012 | Kasuya A, Sawada Y, Tsukamoto Y, Tanaka K, Toya T, Yanagi M: Binding mode of ecdysone agonists to the receptor: comparative modeling and docking studies. J Mol Model. 2003 Feb;9(1):58-65. Epub 2003 Jan 14. Two models were created based both on known ligand-binding domain structures of the receptors with the highest sequence identity to the ecdysone receptor, and on those of steroid hormone receptors. |
2(0,0,0,2) | Details |
8641050 | Kothapalli R, Palli SR, Ladd TR, Sohi SS, Cress D, Dhadialla TS, Tzertzinis G, Retnakaran A: Cloning and developmental expression of the ecdysone receptor gene from the spruce budworm, Choristoneura fumiferana. Dev Genet. 1995;17(4):319-30. Degenerate oligonucleotides were designed on the basis of conserved amino acid sequences in the DNA and ligand-binding regions of the members of the steroid hormone receptor superfamily. |
2(0,0,0,2) | Details |
9131779 | Palli SR, Ladd TR, Retnakaran A: Cloning and characterization of a new isoform of Choristoneura hormone receptor 3 from the spruce budworm. Arch Insect Biochem Physiol. 1997;35(1-2):33-44. |
2(0,0,0,2) | Details |
14503575 | Schneider MI, Smagghe G, Gobbi A, Vinuela E: Toxicity and pharmacokinetics of insect growth regulators and other novel insecticides on pupae of Hyposoter didmator (Hymenoptera: Ichneumonidae), a parasitoid of early larval instars of lepidopteran pests. J Econ Entomol. 2003 Aug;96(4):1054-65. In addition, we tested for the presence of molting hormone receptors in Hyposoter tissues using a monoclonal antibody 9B9. Susceptibility of the lepidopteran parasitoid Hyposoter didymator (Thunberg) to seven modern insecticides, azadirachtin, diflubenzuron, halofenozide, methoxyfenozide, pyriproxyfen, tebufenozide, and spinosad, was tested in the laboratory. |
1(0,0,0,1) | Details |
11755068 | Sundaram M, Palli SR, Smagghe G, Ishaaya I, Feng QL, Primavera M, Tomkins WL, Krell PJ, Retnakaran A: Effect of RH-5992 on adult development in the spruce budworm, Choristoneura fumiferana. Insect Biochem Mol Biol. 2002 Feb;32(2):225-31. The effect of RH-5992 (tebufenozide), a non-steroidal ecdysone agonist, on adult development of the spruce budworm, Choristoneura fumiferana, was investigated by administering the compound intrahemocoelically to pupae on days 1-6 after pupal ecdysis. Injection of RH-5992 into pupae resulted in a dose dependent induction of mRNA for ecdysone-induced transcription factor, Choristoneura hormone receptor 3 (CHR3). |
1(0,0,0,1) | Details |
14745824 | Hu W, Cook BJ, Ampasala DR, Zheng S, Caputo G, Krell PJ, Retnakaran A, Arif BM, Feng Q: Morphological and molecular effects of 20-hydroxyecdysone and its agonist tebufenozide on CF-203, a midgut-derived cell line from the spruce budworm, Choristoneura fumiferana. Arch Insect Biochem Physiol. 2004 Feb;55(2):68-78. The cells responded to these compounds by clumping, generating filamentous extensions, increased mortality and expression of the transcription factor, Choristoneura hormone receptor 3 (CHR3). |
1(0,0,0,1) | Details |
9755479 | Sundaram M, Palli SR, Krell PJ, Sohi SS, Dhadialla TS, Retnakaran A: Basis for selective action of a synthetic molting hormone agonist, RH-5992 on lepidopteran insects. Insect Biochem Mol Biol. 1998 Sep;28(9):693-704. The mRNAs for hormone receptor 3 homologues cloned from Drosophila (DHR3) and Choristoneura (CHR3) are directly induced by 20-hydroxyecdysone (20E) and serve as suitable markers for studying ecdysone action. |
1(0,0,0,1) | Details |
11695189 | Retnakaran A, Gelbic I, Sundaram M, Tomkins W, Ladd T, Primavera M, Feng Q, Arif B, Palli R, Krell P: Mode of action of the ecdysone agonist tebufenozide (RH-5992), and an exclusion mechanism to explain resistance to it. Pest Manag Sci. 2001 Oct;57(10):951-7. |
0(0,0,0,0) | Details |