Protein Information

Name G protein coupled receptor
Synonyms ASRT 2; ASRT2; G protein coupled receptor 154; G protein coupled receptor for asthma susceptibility; G protein coupled receptor; G protein coupled receptor PGR14; GPR154; GPRA…

Compound Information

Name ethylene
CAS ethene

Reference List

PubMed Abstract RScore(About this table)
19785401 Kim Y, Hechler B, Gao ZG, Gachet C, Jacobson KA: PEGylated Dendritic Unimolecular Micelles as Versatile Carriers for Ligands of G Protein-Coupled Receptors. Bioconjug Chem. 2009 Sep 28.

Despite its widespread application in nanomedicine, poly (ethylene glycol) (PEG) is seldom used for covalent modification of ligands for G protein-coupled receptors (GPCRs) due to potential steric complications.
82(1,1,1,2) Details
19475639 Bonger KM, van den Berg RJ, Knijnenburg AD, Heitman LH, van Koppen CJ, Timmers CM, Overkleeft HS, van der Marel GA: Discovery of selective luteinizing hormone receptor agonists using the bivalent ligand method. ChemMedChem. 2009 Jul;4(7):1189-95.


Two series of dimeric ligands for a G-protein-coupled receptor were prepared that differ by the interconnecting spacer system.
2(0,0,0,2) Details