| Name | follicle stimulating hormone receptor |
|---|---|
| Synonyms | FSH R; FSH receptor; FSHR; FSHRO; Follicle stimulating hormone receptor; Follicle stimulating hormone receptor precursor; Follitropin receptor; Follitropin receptor FSHR… |
| Name | ethylene |
|---|---|
| CAS | ethene |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 19902448 | Bonger KM, Hoogendoorn S, van Koppen CJ, Timmers CM, Overkleeft HS, van der Marel GA: Synthesis and pharmacological evaluation of dimeric follicle-stimulating hormone receptor antagonists. ChemMedChem. 2009 Dec;4(12):2098-102. A series of homo- and heterodimeric compounds encompassing the follicle-stimulating hormone receptor (FSHR) antagonist (R)-1 and its inactive conformer (S)-1 connected through ethylene glycol spacers of various lengths is described. |
33(0,1,1,3) | Details |
| 19475639 | Bonger KM, van den Berg RJ, Knijnenburg AD, Heitman LH, van Koppen CJ, Timmers CM, Overkleeft HS, van der Marel GA: Discovery of selective luteinizing hormone receptor agonists using the bivalent ligand method. ChemMedChem. 2009 Jul;4(7):1189-95. Biological evaluation revealed that both dimeric series exhibit unique biological properties relative to their monomeric counterparts.The luteinizing hormone receptor (LHR), the follicle-stimulating hormone receptor (FSHR), and the thyroid-stimulating hormone receptor (TSHR) belong to the glycoprotein hormone receptor (GpHR) family. |
3(0,0,0,3) | Details |