| Name | A2a |
|---|---|
| Synonyms | A2a; A2c; IGKV2D 29; IGKV2D29; immunoglobulin kappa variable 2D 29; A2cs; immunoglobulin kappa variable 2D 29s |
| Name | piperazine |
|---|---|
| CAS | piperazine |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 15294001 | Vu CB, Peng B, Kumaravel G, Smits G, Jin X, Phadke D, Engber T, Huang C, Reilly J, Tam S, Grant D, Hetu G, Chen L, Zhang J, Petter RC: Piperazine derivatives of [1,2,4] triazolo [1,5-a][1,3,5] triazine as potent and selective adenosine A2a receptor antagonists. J Med Chem. 2004 Aug 12;47(17):4291-9. With some preliminary optimization, the A2a binding affinity of some of the best piperazine derivatives is almost as good as that of compound 3. |
81(1,1,1,1) | Details |