| Name | dopamine transporter |
|---|---|
| Synonyms | DA transporter; DAT1; DAT; DAT 1; Dopamine transporter; SLC6A3; Sodium dependent dopamine transporter; Dopamine transporters… |
| Name | diphenylamine |
|---|---|
| CAS |
| PubMed | Abstract | RScore(About this table) | |
|---|---|---|---|
| 10543888 | Husbands SM, Izenwasser S, Kopajtic T, Bowen WD, Vilner BJ, Katz JL, Newman AH: Structure-activity relationships at the monoamine transporters and sigma receptors for a novel series of 9-[3-(cis-3, 5-dimethyl-1-piperazinyl) propyl] carbazole (rimcazole) analogues. J Med Chem. 1999 Oct 21;42(21):4446-55. 9-[3-(cis-3,5-Dimethyl-1-piperazinyl) propyl] carbazole (rimcazole) has been characterized as a sigma receptor antagonist that binds to the dopamine transporter with moderate affinity (K (i) = 224 nM). Analogues in which the carbazole ring was replaced with a freely rotating diphenylamine moiety were also prepared. |
7(0,0,0,7) | Details |
| 15566284 | Cao J, Lever JR, Kopajtic T, Katz JL, Pham AT, Holmes ML, Justice JB, Newman AH: Novel azido and isothiocyanato analogues of [3-(4-phenylalkylpiperazin-1-yl) propyl] bis (4-fluorophenyl) amines as potential irreversible ligands for the dopamine transporter. J Med Chem. 2004 Dec 2;47(25):6128-36. |
1(0,0,0,1) | Details |
| 12742518 | Katz JL, Libby TA, Kopajtic T, Husbands SM, Newman AH: Behavioral effects of rimcazole analogues alone and in combination with cocaine. Eur J Pharmacol. 2003 May 9;468(2):109-19. Several sigma receptor ligands have been reported to also have affinity for the dopamine transporter, among them rimcazole (9-[3-(cis-3,5-dimethyl-1-piperazinyl) propyl] carbazole dihydrochloride). |
1(0,0,0,1) | Details |